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CGRP RECEPTOR ANTAGONISTS
Descriptors Found:
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DeCS
Descriptor
English
:
Calcitonin Gene-Related Peptide Receptor Antagonists
Descriptor
Spanish
:
Antagonistas del Receptor Peptídico Relacionado con el Gen de la Calcitonina
Descriptor
Portuguese
:
Antagonistas do Receptor do Peptídeo Relacionado ao Gene de Calcitonina
Synonyms
English
:
Antagonists, CGRP Receptor
CGRP Receptor Antagonists
Calcitonin Gene Related Peptide Receptor Antagonists
GEPANTS
Receptor Antagonists, CGRP
Tree Number:
D27.505.519.270
D27.505.696.663.850.014.610
D27.505.954.427.040.409
Definition
English
:
Pharmacologic agents that block
NOCICEPTIVE PAIN
signaling from
CALCITONIN GENE-RELATED PEPTIDE
RECEPTORS. They may be useful for the treatment of pain associated with
MIGRAINE DISORDERS
and
OSTEOARTHRITIS.
See Related
English
:
Receptors, Calcitonin Gene-Related Peptide
History Note
English
:
2019
Allowable Qualifiers
English
:
AD
administration & dosage
AE
adverse effects
AN
analysis
BL
blood
CF
cerebrospinal fluid
CS
chemical synthesis
CH
chemistry
CL
classification
EC
economics
HI
history
IM
immunology
IP
isolation & purification
ME
metabolism
PK
pharmacokinetics
PD
pharmacology
PO
poisoning
RE
radiation effects
ST
standards
SD
supply & distribution
TU
therapeutic use
TO
toxicity
UR
urine
Record Number:
57552
Unique Identifier:
D000077221
Occurrence in VHL
:
Similar:
DeCS